Timeline

26 Jan 2021

publication

Core-Modified Coelenterazine Luciferin Analogues: Synthesis and Chemiluminescence Properties.

12 Jan 2021

publication

Measuring the subcellular compartmentalization of viral infections by protein complementation assay.

01 Jan 2021

publication

High seroprevalence but short-lived immune response to SARS-CoV-2 infection in Paris.

01 Nov 2020

publication

A highly sensitive bioluminescent method for measuring allergen-specific IgE in microliter samples.

12 Feb 2020

event

Department of Structural Biology and Chemistry: Bernard Meunier, Que d’échecs dans la recherche de médicaments pour traiter la maladie d’Alzheimer !

16 Jan 2020

publication

Bioluminescence Profiling of NanoKAZ/NanoLuc Luciferase Using a Chemical Library of Coelenterazine Analogues.

12 Nov 2019

event

Molecular basis for evolution of the Renilla-type bioluminescence

29 Aug 2019

publication

Maximizing binary interactome mapping with a minimal number of assays

15 Jul 2019

event

Department of Structural Biology & Chemistry seminar: Dr. Bernard Meunier, Que d’échecs dans la recherche de médicaments pour traiter la maladie d’Alzheimer !

10 Apr 2019

publication

Gram-scale synthesis of luciferins derived from coelenterazine and original insights into their bioluminescence properties.

16 Nov 2018

publication

Unnatural α-amino ethyl esters from diethyl malonate or ethyl β-bromo-α-hydroxyiminocarboxylate

15 Nov 2018

publication

Synthesis of unnatural α-amino esters using ethyl nitroacetate and condensation or cycloaddition reactions

10 Aug 2017

publication

Synthesis of α-Amino Esters via α-Nitro or α-Oxime Esters: A Review

12 Jul 2017

publication

Checkpoint kinase 1 inhibition sensitises transformed cells to dihydroorotate dehydrogenase inhibition

25 Sep 2015

publication

Synthetic Routes to Coelenterazine and Other Imidazo[1,2-a]pyrazin-3-one Luciferins: Essential Tools for Bioluminescence-Based Investigations

18 Aug 2015

project

Design and optimization of new bioluminescent systems better-suited to in cellulo and in vivo conditions

28 Jul 2015

project

Alkoxypyrazoles, inhibitors of dihydroorotate dehydrogenase (DHODH)

24 Jul 2015

project

Alkoxypyrazoles, new chemical entities

30 Jun 2015

publication

Original 2-(3-Alkoxy-1H-pyrazol-1-yl)azines Inhibitors of Human Dihydroorotate Dehydrogenase (DHODH)

10 Feb 2015

publication

A study of Negishi cross-coupling reactions with benzylzinc halides to prepare original 3-ethoxypyrazoles

06 Jan 2015

publication

Original 2-(3-alkoxy-1H-pyrazol-1-yl)pyrimidine derivatives as inhibitors of human dihydroorotate dehydrogenase (DHODH)

20 Mar 2013

publication

On dihydroorotate dehydrogenases and their inhibitors and uses

01 Jan 2013

publication

Pyrazole-3/5-carboxylic acids from 3/5-trifluoromethyl NH-pyrazoles

01 Jan 2013

publication

Preparations of 4-subtituted 3-carboxypyrazoles

01 May 2012

publication

Preparation and chemistry of 3/5-halogenopyrazoles

01 Jan 2012

publication

3-Methoxypyrazoles from 1,1-dimethoxyethene, few original results

01 Jan 2012

publication

Few unexpected results from a Suzuki-Miyaura reaction

01 Jan 2011

publication

On the Knorr synthesis of 6-bromo-4-methylquinolin-2(1H)-one

01 Jan 2011

publication

Simple preparations of 4 and 5-iodinated pyrazoles as useful building blocks

01 Oct 2010

publication

Synthesis, biological activity, and evaluation of the mode of action of novel antitubercular benzofurobenzopyrans substituted on A ring

23 Mar 2010

publication

5-Iodo-3-ethoxypyrazoles: an entry point to new chemical entities

15 Mar 2010

publication

ATPase inhibitors of heat-shock protein 90, second season

01 Jan 2010

publication

Synthetic accesses to 3/5-pyrazole carboxylic acids

01 Jan 2010

publication

N-arylation of 3-alkoxypyrazoles, the case of the pyridines

29 Jan 2009

publication

Diversity-oriented synthesis of furo[3,2-f]chromanes with antimycobacterial activity

01 Jan 2009

publication

Carbon-4 arylation of 3-alkoxypyrazoles

01 Jan 2009

publication

Nitrogen’s reactivity of various 3-alkoxypyrazoles

03 Aug 2008

publication

A new synthetic access to furo[3,2-f]chromene analogues of an antimycobacterial

01 Jan 2008

publication

An improved preparation of 3-alkoxypyrazoles

01 Jan 2008

publication

Optimized palladium-based approaches to analogues of PK 11195

19 Jan 2007

publication

Antituberculosis drugs: ten years of research

01 Jan 2007

publication

Isoxyl activation is required for bacteriostatic activity against Mycobacterium tuberculosis

01 Jan 2007

publication

Antimycobacterial benzofuro[3,2-f]chromenes from a 5-bromochromen-6-ol

12 Dec 2006

publication

Synthesis and antimycobacterial evaluation of benzofurobenzopyran analogues

01 Jan 2006

publication

A simple two steps ytterbium triflate-catalysed preparation of 2,2-dimethylchromenes from salicylaldehydes and 2-methylpropene

01 Dec 2005

publication

Heat shock protein 90 inhibitors. A text book example of medicinal chemistry?

01 Jan 2004

publication

Synthesis of methylenedioxy-bearing 1-aryl-3-carboxylisoquinolines using a modified Ritter reaction procedure

01 Jan 2003

publication

Peptides with anticancer use or potential

01 Jul 2002

publication

A little guide for advanced search:

Core-Modified Coelenterazine Luciferin Analogues: Synthesis and Chemiluminescence Properties.

Measuring the subcellular compartmentalization of viral infections by protein complementation assay.

High seroprevalence but short-lived immune response to SARS-CoV-2 infection in Paris.

A highly sensitive bioluminescent method for measuring allergen-specific IgE in microliter samples.

Department of Structural Biology and Chemistry: Bernard Meunier, Que d’échecs dans la recherche de médicaments pour traiter la maladie d’Alzheimer !

Bioluminescence Profiling of NanoKAZ/NanoLuc Luciferase Using a Chemical Library of Coelenterazine Analogues.

Molecular basis for evolution of the Renilla-type bioluminescence

Maximizing binary interactome mapping with a minimal number of assays

Department of Structural Biology & Chemistry seminar: Dr. Bernard Meunier, Que d’échecs dans la recherche de médicaments pour traiter la maladie d’Alzheimer !

Gram-scale synthesis of luciferins derived from coelenterazine and original insights into their bioluminescence properties.

Unnatural α-amino ethyl esters from diethyl malonate or ethyl β-bromo-α-hydroxyiminocarboxylate

Synthesis of unnatural α-amino esters using ethyl nitroacetate and condensation or cycloaddition reactions

Synthesis of α-Amino Esters via α-Nitro or α-Oxime Esters: A Review

Checkpoint kinase 1 inhibition sensitises transformed cells to dihydroorotate dehydrogenase inhibition

Synthetic Routes to Coelenterazine and Other Imidazo[1,2-a]pyrazin-3-one Luciferins: Essential Tools for Bioluminescence-Based Investigations

Design and optimization of new bioluminescent systems better-suited to in cellulo and in vivo conditions

Alkoxypyrazoles, inhibitors of dihydroorotate dehydrogenase (DHODH)

Alkoxypyrazoles, new chemical entities

Original 2-(3-Alkoxy-1H-pyrazol-1-yl)azines Inhibitors of Human Dihydroorotate Dehydrogenase (DHODH)

A study of Negishi cross-coupling reactions with benzylzinc halides to prepare original 3-ethoxypyrazoles

Original 2-(3-alkoxy-1H-pyrazol-1-yl)pyrimidine derivatives as inhibitors of human dihydroorotate dehydrogenase (DHODH)

On dihydroorotate dehydrogenases and their inhibitors and uses

Pyrazole-3/5-carboxylic acids from 3/5-trifluoromethyl NH-pyrazoles

Preparations of 4-subtituted 3-carboxypyrazoles

Preparation and chemistry of 3/5-halogenopyrazoles

3-Methoxypyrazoles from 1,1-dimethoxyethene, few original results

Few unexpected results from a Suzuki-Miyaura reaction

On the Knorr synthesis of 6-bromo-4-methylquinolin-2(1H)-one

Simple preparations of 4 and 5-iodinated pyrazoles as useful building blocks

Synthesis, biological activity, and evaluation of the mode of action of novel antitubercular benzofurobenzopyrans substituted on A ring

5-Iodo-3-ethoxypyrazoles: an entry point to new chemical entities

ATPase inhibitors of heat-shock protein 90, second season

Synthetic accesses to 3/5-pyrazole carboxylic acids

N-arylation of 3-alkoxypyrazoles, the case of the pyridines

Diversity-oriented synthesis of furo[3,2-f]chromanes with antimycobacterial activity

Carbon-4 arylation of 3-alkoxypyrazoles

Nitrogen’s reactivity of various 3-alkoxypyrazoles

A new synthetic access to furo[3,2-f]chromene analogues of an antimycobacterial

An improved preparation of 3-alkoxypyrazoles

Optimized palladium-based approaches to analogues of PK 11195

Antituberculosis drugs: ten years of research

Isoxyl activation is required for bacteriostatic activity against Mycobacterium tuberculosis

Antimycobacterial benzofuro[3,2-f]chromenes from a 5-bromochromen-6-ol

Synthesis and antimycobacterial evaluation of benzofurobenzopyran analogues

A simple two steps ytterbium triflate-catalysed preparation of 2,2-dimethylchromenes from salicylaldehydes and 2-methylpropene

Heat shock protein 90 inhibitors. A text book example of medicinal chemistry?

Synthesis of methylenedioxy-bearing 1-aryl-3-carboxylisoquinolines using a modified Ritter reaction procedure

Peptides with anticancer use or potential

2-Amino-3-(3-hydroxy-1,2,5-thiadiazol-4-yl)propionic acid: resolution, absolute stereochemistry and enantiopharmacology at glutamate receptors