Timeline
Ludovic Halby
Research Engineer
22 May 2023
publication
Plasmodium falciparum Eukaryotic Translation Initiation Factor 3 is Stabilized by Quinazoline-Quinoline Bisubstrate Inhibitors.
Read more17 Feb 2023
publication
Hemisynthetic alkaloids derived from trilobine are antimalarials with sustained activity in multidrug-resistant Plasmodium falciparum.
Read more11 Jan 2023
news
New publication: Hemisynthetic alkaloids derived from trilobine are antimalarials with sustained activity in multidrug-resistant Plasmodium falciparum
Read more01 Apr 2022
publication
Quinazoline-based analog of adenine as an antidote against MLL-rearranged leukemia cells: synthesis, inhibition assays and docking studies.
Read more01 Dec 2021
publication
Direct Synthesis of Allyl Amines with 2-Nitrosulfonamide Derivatives via the Tsuji-Trost Reaction.
Read more31 Aug 2021
publication
Synthesis and Biological Activity of a Cytostatic Inhibitor of MLLr Leukemia Targeting the DOT1L Protein
Read more15 Aug 2021
publication
Direct Synthesis of Allyl Amines with 2‐Nitrosulfonamide Derivatives via the Tsuji‐Trost Reaction
Read more22 Jul 2021
publication
Procainamide-SAHA Fused Inhibitors of hHDAC6 Tackle Multidrug-Resistant Malaria Parasites.
Read more18 Feb 2021
project
Epi-Med: synthesis and biological evaluation of new active molecules against MLL-rearranged leukaemia.
Read more18 Feb 2021
project
EpiKillMal- Use of DNA methyltransferase inhibitors to kill drug-resistant malaria parasites –
Read more17 Sep 2020
publication
Bisubstrate inhibitors: the promise of a selective and potent chemical inhibition of epigenetic ‘writers’
Read more01 Sep 2020
publication
Bisubstrate inhibitors: the promise of a selective and potent chemical inhibition of epigenetic ‘writers’.
Read more19 Mar 2020
publication
Bisubstrate-Type Chemical Probes Identify GRP94 as a Potential Target of Cytosine-Containing Adenosine Analogs.
Read more22 Jan 2020
publication
DNA Methylation Bisubstrate Inhibitors Are Fast-Acting Drugs Active against Artemisinin-Resistant Plasmodium falciparum Parasites.
Read more01 Oct 2019
publication
[Chemical targeting of DNA and histone methylation in cancer: Novelties, hopes and promises].
Read more24 Sep 2019
19 Sep 2019
publication
Espoirs et promesses de la méthylation de l’ADN et des histones comme cibles anticancéreuses
Read more09 Jan 2018