Ligne de temps
Ludovic Halby
Ingénieur(e) de Recherche
22 mai 2023
publication
Plasmodium falciparum Eukaryotic Translation Initiation Factor 3 is Stabilized by Quinazoline-Quinoline Bisubstrate Inhibitors.
Lire plus17 févr. 2023
publication
Hemisynthetic alkaloids derived from trilobine are antimalarials with sustained activity in multidrug-resistant Plasmodium falciparum.
Lire plus11 janv. 2023
news
New publication: Hemisynthetic alkaloids derived from trilobine are antimalarials with sustained activity in multidrug-resistant Plasmodium falciparum
Lire plus01 avr. 2022
publication
Quinazoline-based analog of adenine as an antidote against MLL-rearranged leukemia cells: synthesis, inhibition assays and docking studies.
Lire plus01 déc. 2021
publication
Direct Synthesis of Allyl Amines with 2-Nitrosulfonamide Derivatives via the Tsuji-Trost Reaction.
Lire plus31 août 2021
publication
Synthesis and Biological Activity of a Cytostatic Inhibitor of MLLr Leukemia Targeting the DOT1L Protein
Lire plus15 août 2021
publication
Direct Synthesis of Allyl Amines with 2‐Nitrosulfonamide Derivatives via the Tsuji‐Trost Reaction
Lire plus22 juil. 2021
publication
Procainamide-SAHA Fused Inhibitors of hHDAC6 Tackle Multidrug-Resistant Malaria Parasites.
Lire plus18 févr. 2021
project
Epi-Med: synthesis and biological evaluation of new active molecules against MLL-rearranged leukaemia.
Lire plus18 févr. 2021
project
EpiKillMal- Use of DNA methyltransferase inhibitors to kill drug-resistant malaria parasites –
Lire plus17 sept. 2020
publication
Bisubstrate inhibitors: the promise of a selective and potent chemical inhibition of epigenetic ‘writers’
Lire plus01 sept. 2020
publication
Bisubstrate inhibitors: the promise of a selective and potent chemical inhibition of epigenetic ‘writers’.
Lire plus19 mars 2020
publication
Bisubstrate-Type Chemical Probes Identify GRP94 as a Potential Target of Cytosine-Containing Adenosine Analogs.
Lire plus22 janv. 2020
publication
DNA Methylation Bisubstrate Inhibitors Are Fast-Acting Drugs Active against Artemisinin-Resistant Plasmodium falciparum Parasites.
Lire plus01 oct. 2019
publication
[Chemical targeting of DNA and histone methylation in cancer: Novelties, hopes and promises].
Lire plus24 sept. 2019
19 sept. 2019
publication
Espoirs et promesses de la méthylation de l’ADN et des histones comme cibles anticancéreuses
Lire plus09 janv. 2018