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2021Core-Modified Coelenterazine Luciferin Analogues: Synthesis and Chemiluminescence Properties., Chemistry 2021 Jan; 27(6): 2112-2123.
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2021Measuring the subcellular compartmentalization of viral infections by protein complementation assay., Proc Natl Acad Sci U S A 2021 01; 118(2): .
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2021High seroprevalence but short-lived immune response to SARS-CoV-2 infection in Paris., Eur J Immunol 2021 01; 51(1): 180-190.
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2020A highly sensitive bioluminescent method for measuring allergen-specific IgE in microliter samples., Allergy 2020 11; 75(11): 2952-2956.
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2020Bioluminescence Profiling of NanoKAZ/NanoLuc Luciferase Using a Chemical Library of Coelenterazine Analogues., Chemistry 2020 Jan; 26(4): 948-958.
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2019Maximizing binary interactome mapping with a minimal number of assays, Nat Commun 2019 Aug;10(1):3907.
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2019Gram-scale synthesis of luciferins derived from coelenterazine and original insights into their bioluminescence properties., Org Biomol Chem 2019 04; 17(15): 3709-3713.
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2018Unnatural α-amino ethyl esters from diethyl malonate or ethyl β-bromo-α-hydroxyiminocarboxylate, Beilstein J Org Chem 2018;14:2853-2860.
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2018Synthesis of unnatural α-amino esters using ethyl nitroacetate and condensation or cycloaddition reactions, Beilstein J Org Chem 2018;14:2846-2852.
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2017Synthesis of α-Amino Esters via α-Nitro or α-Oxime Esters: A Review, Synthesis 2017, DOI: 10.1055/s-0036-1589506.
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2017Checkpoint kinase 1 inhibition sensitises transformed cells to dihydroorotate dehydrogenase inhibition, Oncotarget 2017 Jul;.
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2015Synthetic Routes to Coelenterazine and Other Imidazo[1,2-a]pyrazin-3-one Luciferins: Essential Tools for Bioluminescence-Based Investigations, Chemistry 2015 Nov;21(48):17158-71.
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2015Original 2-(3-Alkoxy-1H-pyrazol-1-yl)azines Inhibitors of Human Dihydroorotate Dehydrogenase (DHODH), J. Med. Chem. 2015 Jul;58(14):5579-98.
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2015A study of Negishi cross-coupling reactions with benzylzinc halides to prepare original 3-ethoxypyrazoles, Synthesis 2015, 47, 511-516.
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2015Original 2-(3-alkoxy-1H-pyrazol-1-yl)pyrimidine derivatives as inhibitors of human dihydroorotate dehydrogenase (DHODH), J. Med. Chem. 2015 Jan;58(2):860-77.
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2013On dihydroorotate dehydrogenases and their inhibitors and uses, J. Med. Chem. 2013 Apr;56(8):3148-67.
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2013Pyrazole-3/5-carboxylic acids from 3/5-trifluoromethyl NH-pyrazoles, Tetrahedron 2013, 69, 257-263.
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2013Preparations of 4-subtituted 3-carboxypyrazoles, J. Heterocycl. Chem. 2013, 50, 1410-1414.
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2012Preparation and chemistry of 3/5-halogenopyrazoles, Chem. Rev. 2012 Jul;112(7):3924-58.
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20123-Methoxypyrazoles from 1,1-dimethoxyethene, few original results, Tetrahedron 2012, 68, 3165-3171.
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2012Few unexpected results from a Suzuki-Miyaura reaction, Tetrahedron 2012, 68, 2135-2140.
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2011On the Knorr synthesis of 6-bromo-4-methylquinolin-2(1H)-one, Synthesis 2011, (6), 934-942.
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2011Simple preparations of 4 and 5-iodinated pyrazoles as useful building blocks, Tetrahedron 2011, 67, 8451-8457.
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2010Synthesis, biological activity, and evaluation of the mode of action of novel antitubercular benzofurobenzopyrans substituted on A ring, Eur J Med Chem 2010 Dec;45(12):5833-47.
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20105-Iodo-3-ethoxypyrazoles: an entry point to new chemical entities, Chemistry 2010 Apr;16(15):4669-77.
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2010ATPase inhibitors of heat-shock protein 90, second season, Drug Discov. Today 2010 May;15(9-10):342-53.
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2010Synthetic accesses to 3/5-pyrazole carboxylic acids, Mini Rev. Org. Chem. 2010, 7, 314-323.
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2010N-arylation of 3-alkoxypyrazoles, the case of the pyridines, Tetrahedron 2010, 66, 2654-2663.
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2009Diversity-oriented synthesis of furo[3,2-f]chromanes with antimycobacterial activity, Eur J Med Chem 2009 Jun;44(6):2497-505.
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2009Carbon-4 arylation of 3-alkoxypyrazoles, Tetrahedron 2009, 65, 3529-3535.
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2009Nitrogen’s reactivity of various 3-alkoxypyrazoles, Tetrahedron 2009, 65, 2660-2668.
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2008A new synthetic access to furo[3,2-f]chromene analogues of an antimycobacterial, Bioorg. Med. Chem. 2008 Sep;16(17):8264-72.
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2008Optimized palladium-based approaches to analogues of PK 11195, J. Heterocycl. Chem. 2008, 45, 1377-1384.
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2008An improved preparation of 3-alkoxypyrazoles, Synthesis 2008, 3504-3508.
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2007Antituberculosis drugs: ten years of research, Bioorg. Med. Chem. 2007 Apr;15(7):2479-513.
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2007Isoxyl activation is required for bacteriostatic activity against Mycobacterium tuberculosis, Antimicrob. Agents Chemother. 2007, 51, 3824-3829.
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2007Antimycobacterial benzofuro[3,2-f]chromenes from a 5-bromochromen-6-ol, Synthesis 2007, 1566-1570.
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2006Synthesis and antimycobacterial evaluation of benzofurobenzopyran analogues, Bioorg. Med. Chem. 2007 Mar;15(5):2177-86.
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2006A simple two steps ytterbium triflate-catalysed preparation of 2,2-dimethylchromenes from salicylaldehydes and 2-methylpropene, J. Heterocycl. Chem. 2006, 43, 1605-1608.
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2005Heat shock protein 90 inhibitors. A text book example of medicinal chemistry?, J. Med. Chem. 2005 Dec;48(24):7503-12.
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2004Synthesis of methylenedioxy-bearing 1-aryl-3-carboxylisoquinolines using a modified Ritter reaction procedure, Tetrahedron 2004, 60, 5481-5485.
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2003Peptides with anticancer use or potential, Amino Acids 2003, 25, 1-40.
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20022-Amino-3-(3-hydroxy-1,2,5-thiadiazol-4-yl)propionic acid: resolution, absolute stereochemistry and enantiopharmacology at glutamate receptors, Bioorg. Med. Chem. 2002 Jul;10(7):2259-66.